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AbMole丨铜离子载体Elesclomol(STA-4783):靶向线粒体诱导铜死亡
Elesclomol(STA-4783,AbMole,M2083)是一种线粒体靶向小分子化合物,核心机制在于作为铜离子载体(Cu²⁺ ionophore),与外源铜离子形成复合物(Elesclomol-Cu),将铜高效转运至线粒体基质,触发铜依赖性细胞死亡--铜死亡(Cuproptosis)。上述过程依赖于线粒体还原 ...
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