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AbMole丨Wortmannin(渥曼青霉素):强效PI3K家族抑制剂,在信号转导 ...
Wortmannin(渥曼青霉素,AbMole,M2053)是一种源自真菌的甾体代谢物,作为磷脂酰肌醇3-激酶(PI3K)家族的强效共价抑制剂,能不可逆地结合PI3K催化亚基。Wortmannin还能抑制同属PI3K家族的DNA依赖性蛋白激酶(DNA-PK)和共济失调毛细血管扩张症突变激酶(ATM)。在生物学活性上,Wortmannin(渥曼青霉素,AbMole,M2053) ...
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